Recettori nucleari per ormoni steroidei

A receptor which is capable of producing a biological response in the absence of a bound ligand is said to display "constitutive activity". [5] The constitutive activity of a receptor may be blocked by an inverse agonist . The anti-obesity drugs rimonabant and taranabant are inverse agonists at the cannabinoid CB1 receptor and though they produced significant weight loss, both were withdrawn owing to a high incidence of depression and anxiety, which are believed to relate to the inhibition of the constitutive activity of the cannabinoid receptor.

Recettori nucleari per ormoni steroidei

recettori nucleari per ormoni steroidei

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recettori nucleari per ormoni steroideirecettori nucleari per ormoni steroideirecettori nucleari per ormoni steroideirecettori nucleari per ormoni steroideirecettori nucleari per ormoni steroidei